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Top 100 Small-Molecule Drugs by US Retail Sales in 2012

1
Jan
1

13

NexIUM

Modified from the list produced by the Njardarson Group (The University of Arizona)

2
Feb
2

Abilify

3
Mar
3

Crestor

Advair Diskus

6
Jun

5
May

4
Apr

Cymbalta

Singulair*

11

Januvia

12

Truvada

( Duloxetine )

( Montelukast )

( Clopidogrel )

( Emtricitabine, Tenofovir Disoproxil & Efavirenz )

( Tiotropium )

( Oxycodone )

( Sitagliptin )

( Emtricitabine & Tenofovir )

$5,989 Million
ANTIULCERANTS

$5,870 Million

$5,092 Million

$4,889 Million
CORTICOIDS

$4,720 Million

$3,300 Million

$2,971 Million

$2,899 Million
HIV ANTIVIRALS

$2,833 Million

$2,808 Million

$2,670 Million

$2,305 Million
HIV ANTIVIRALS

Diovan

14

Lyrica

15

( Pregabelin )

Lipitor

Celebrex

16

17

( Atorvastatin )

Gleevec

Namenda

18

( Imatinib )

( Celecoxib )

26

ProAir HFA

38

Incivek

27

Diovan HCT

( Telaprevir )

( Valsartan & Hydrochlorothiazide )

ANTIVIRAL

ANGIOTEN-II ANTAG, COMB

Niaspan

39

( Niacin )

Nasonex

Lidoderm

28

29

( Lidocaine )

Lovaza

40

41

Omega 3-Acid Ethyl Esters )

( Mometasone )

Adderall XR

50

51

( Ciclosporine )

( Amphetamine & Dextroamphetamine )

Synthroid

Restasis

62

Atorvastatin

52

63

Xeloda

74

( Daptomycin )

Detrol LA
( Tolterodine )

Zometa

86

( Mesalazine )

Bystolic

87

Viread*

88

( Tenofovir )

( Nebivolol )

( Amphetamine & Dextroamphetamine )

98

99
( Escitalopram )

Provigil

Vytorin

Colcrys

54

VESIcare

55

( Solifenacin )

Dexilant*

66

Velcade

67

( Bortezomib )

78

Solodyn

Sensipar
( Cinacalcet )

79

Escitalopram
( Escitalopram )

ANTICANCER

ANTIARTHRITIS

ANTIBIOTIC

ANTIDEPRESS.& MOOD STAB.

89

Loestrin 24 Fe

( Norethindrone Acetate & Ethinyl Estradiol )

32

Suboxone

22

33

Alimta

34

( Pemetrexed )

44

Isentress

45

Eloxatin

Budesonide

46

Janumet

90

Avodart

91

Lexiscan

Zetia

24
( Methylphenidate )

( Ezetimibe )

35

( Oxaliplatin )

( Budesonide )

( Raltegravir )

23

( Quetiapine )

( Buprenorphine & Naloxone )

Tricor

SEROquel

Combivent

36

Viagra

48

AcipHex

( Salbutamol & Ipratropium )

47

Cialis

( Rabeprazole )

( Sitagliptin & Metformin )

ANTIULCERANTS

56

57

Lexapro
( Escitalopram )

58

Benicar

Lunesta

59

( Eszopiclone )

( Olmesartan )

ANTIULCERANTS

( Minocycline )

Enoxaparin

21
( Lisdexamfetamine )

( Dexlansoprazole )

( Colchicine )

( Enoxaparin )

100

43

( Bendamustine )

HIV ANTIVIRALS

97

Ventolin HFA

B2-STIMULANTS

ANTIBACTERIAL

Asacol

Prezista

20

( Quetiapine )

LIP.REG.CO.W.OTH.LIP.REG

OTHER ANTIBACTERIALS

( Zolendronic Acid )

Reyataz

SEROquel XR

HIV ANTIVIRALS

HIV ANTIVIRALS

77

31

CORTICOIDS

MULTIPLE SCLEROSIS

Treanda

GLITAZONE ANTIDIABETICS

( Ezetimibe & Simvastatin )

( Salbutamol )

76

ANTI-ALZHEIMER

( Atazanavir )

( Darunavir )

65

( Pioglitazone )

( Budesonide & Formoterol )

42

ACTOS

( Memantine )

Symbicort

30

19

( Fluticasone Propionate )

( Linezolid )

( Capecitabine )

75

53

Flovent HFA

( Fingolimod )

Zyvox

64

ANTIARTHRITIC

Cubicin

Gilenya

( Dabigatran )

( Atorvastatin )

( Levothyroxine )

Pradaxa

Atorvastatin
( Atorvastatin )

B2-STIMULANTS

85

10

Atripla

( Fluticasone Propionate )

( Salbutamol )

73

12
Dec

11
Nov

( Rosuvastatin )

25

61

Plavix

10
Oct

( Aripiprazole )

ANTIEPILEPTICS

49

9
Sep

( Esomeprazole )

( Valsartan )

37

8
Aug

7
Jul

68

Pristiq

70

( Ocreotide Acetate )

( Olmesartan & Hydrochlorothiazide )

80

69

81

Invega Sustenna

71

82

Strattera

60

83

Enoxaparin

( Raloxifene )

( Enoxaparin )

SERMS

HUMAN INSULIN+ANALOGUES

Focalin XR

72

( Dexmethylphenidate )

( Levonorgestrel )

( Paliperidone Palmitate )

( Desvenlafaxine )

Mirena

Evista

Trilipix

Tarceva
( Erlotinib )

84

( Atomoxetine )

Revlimid
( Lenalidomide )

ANTIPSYCHOTIC

92

Lovenox

93

Epzicom*

( Dutasteride )

( Regadenoson )

( Enoxaparin )

( Abacavir & Lamivudine )

BPH PRODUCTS

CORONARY VASODILATOR

HEPARINS

HIV ANTIVIRALS

94

95
( Rivastigmine )

96

( Amphetamine & Dextroamphetamine )

( Etonogestrel & Ethinyl Estradiol )

Norvir
( Ritonavir )

*Modified chemical structures from original version

HIV ANTIVIRAL

Reference
http://www.pharmacytimes.com/publications/issue/2013/July2013/Top-200-Drugs-of-2012

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