Beruflich Dokumente
Kultur Dokumente
p-Blockers
257
Drug
NONSELECTIVE
propranolol (Inderal)
nadolol (Corgard)
penbutolol (Levatol)
pindolol (Visken)
sotalol (Betapace, Betapace AF)
Hypertension
Angina
CHF
/
/
Arrhythmias
ISA
Other Uses
Migraineprophylaxis, essen
tialtremor, hypertrophic
subaortic stenosis, pheo-
chromocytoma, Graves'
disease. Ml prophylaxis
/
/
timolol (Blocadren)
Migraine prophylaxis
p,-SELECTIVE
atenolol (Tenormin)
metoprolol (Lopressor,
Toprol XL)
acebutolol (Sectral)
betaxolol (Kerlone)
/ (extended-
releaseonly)
Glaucoma
bisoprolol (Zebeta)
esmolol (Brevibloc) (IV
only)
a-p-BLOCKER
nebivolol (Bystolic)
labetalol (Normodyne,
/
/
Ml prophylaxis, acute Ml
Ml prophylaxis, acute Ml
Trandate)
carvedilol (Coreg)
TABLE 20-2
Receptor
a,
Site
Effect of Stimulation
Vasoconstriction
vessels
0.2
Stomach, intestine
Kidney
Liver
Gluconeogenesis
Vasodilation
vessels
Pi
Cardiac
P2
Kidney
Vasodilation
Decreased secretion
Liver
Gluconeogenesis