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Increase HR (large

doses), decrease HR
(small doses)

Bronchodialation,
decrease secretions

Relaxation of smooth
Contraction of pupils,
muscle tone, motility,
bronchioles
peristalsis, gastric
secretions
Increase bronchial
secretions
Relaxation of detrusor
Effects muscle
Decreased HR

Spincter constriction
Effects
Vasodilation

Dilation of pupils,
decreased
Increased peristalsis,
accommodation
gastric secretions,
salivation

Decreased salivation,
perspiration
Bladder muscle
contraction
Agonist Cholinergic Antagonist Decrease termors,
rigidity of muslces
Smooth muscles (GI,
Decreases HR, glands, lungs, bladder), Muscarinic
heart, eyes
Smooth muscles (GI,
Receptors
Muscarinic glands, lungs, bladder),
heart, eyes
Skeletal muscles Nicotinic
Receptors

Skeletal muscles /
Muscarinic Direct-acting Nicotinic
contraction
Drugs

Muscarinic, nicotinic Indirect-acting


Atropine muscarinic (selective)

Drugs

Benztropine muscarinic (selective)

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